SCHEMBL9243104

SCHEMBL9243104

COc1ccccc1C1(O)CCC(c2ccccc2)(c2ccccc2)[C@H]2CN(C(=O)Cc3c[nH]c4ccc(F)cc34)CC21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.55
FNTA P49354 6/20 0.47
FNTB P49356 6/20 0.47
OPRK1 P41145 1/20 0.45
ICMT O60725 1/20 0.43
TSHR P16473 2/20 0.42
HSD11B1 P28845 1/20 0.41
HTR1A P08908 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR7 P34969 1/20 0.41
KCNH2 Q12809 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8956827 1.00 TACR1 (0.55) TACR1FNTAFNTBOPRK1ICMT
SCHEMBL9245521 0.93 TACR1 (0.54) TACR1FNTAFNTBOPRK1ICMT
SCHEMBL8957016 0.93 TACR1 (0.54) TACR1FNTAFNTBOPRK1ICMT
SCHEMBL8956847 0.92 TACR1 (0.58) TACR1FNTAFNTBOPRK1TSHR
SCHEMBL8956681 0.92 TACR1 (0.58) TACR1FNTAFNTBOPRK1TSHR
SCHEMBL8895210 0.88 FNTA (0.44) TACR1FNTAFNTBOPRK1ICMT
SCHEMBL8545840 0.84 TACR1 (0.67) TACR1FNTAFNTBTSHRMEN1
SCHEMBL8956909 0.84 TACR1 (0.67) TACR1FNTAFNTBTSHRMEN1
SCHEMBL8873453 0.82 OPRK1 (0.48) TACR1FNTAFNTBOPRK1ICMT
SCHEMBL8548669 0.81 TACR1 (0.64) TACR1FNTAFNTBOPRK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463077-A Exhibit substance P antagonist activity RHONE-POULENC RORER S.A. (FR) 1995-10-31 US disclosed