SCHEMBL8957140

SCHEMBL8957140

N[C@@H](Cc1cnc(Cc2ccccc2)[nH]1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.54
ALPI P09923 1/20 0.54
PKM P14618 1/20 0.54
PTGS1 P23219 1/20 0.54
XIAP P98170 1/20 0.54
CYP3A4 P08684 1/20 0.47
BRS3 P32247 2/20 0.45
AOC3 Q16853 1/20 0.45
SLC1A3 P43003 2/20 0.45
SLC1A2 P43004 2/20 0.45
SLC1A1 P43005 2/20 0.45
HSD17B10 Q99714 1/20 0.43
HPGDS O60760 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10584263 0.80 SLC7A5 (0.58) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL28526629 0.79 SLC7A5 (0.47) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL28938740 0.79 SLC7A5 (0.47) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL27446953 0.79 SLC7A5 (0.51) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL29356218 0.79 SLC7A5 (0.51) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7345076 0.79 BRS3 (0.49) BRS3AOC3HPGDS
SCHEMBL849758 0.79 SLC7A5 (0.51) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL9314265 0.78 KEAP1 (0.50) BRS3AOC3HSD17B10HPGDS
SCHEMBL5292853 0.77 SLC7A5 (0.53) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL1539194 0.77 SLC7A5 (0.53) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113924290-A Thiohydrazinocarboxylic acid esters and their use 范因斯坦医学研究院 2022-01-11 CN disclosed
US-5565480-A ANGIOTENSIN II RECEPTOR ANTAGONIST; USEFUL IN REGULATING HYPERTENSION, TREATMENT OF CONGESTIVE HEART FAILURE, RENAL FAILURE AND GLUCOMA SMITHKLINE BEECHAM CORPORATION (US) 1996-10-15 US disclosed
EP-0536262-A4 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORP (US) 1996-08-14 EP disclosed
US-5444081-A Treatment of hypertension, congestive heart failure, renal failure, glaucoma SMITHKLINE BEECHAM CORP (US) 1995-08-22 US disclosed
EP-0536262-A1 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-14 EP disclosed
WO-1992000068-A1 SUBSTITUTED HISTIDINES SMITHKLINE BEECHAM CORPORATION (US) 1992-01-09 WO disclosed