SCHEMBL8958229

SCHEMBL8958229

CC(C)(C)OC(=O)c1ccccc1-c1ccc(CNC(=O)C2(N)CCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.51
BDKRB1 P46663 2/20 0.48
LTB4R2 Q9NPC1 1/20 0.41
SCN9A Q15858 6/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
SLC6A3 Q01959 3/20 0.38
SLC6A4 P31645 2/20 0.38
BRS3 P32247 1/20 0.38
HDAC1 Q13547 1/20 0.38
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
AGTR1 P30556 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8958363 0.91 BDKRB1 (0.46) ACHEBDKRB1LTB4R2SCN9ACHRNB2
SCHEMBL9447504 0.86 ACHE (0.49) ACHEBDKRB1LTB4R2SLC6A3SLC6A4
SCHEMBL5782374 0.84 BDKRB1 (0.60) ACHEBDKRB1LTB4R2CHRNB2CHRNB4
SCHEMBL9032066 0.79 GAA (0.48) ACHEBDKRB1LTB4R2CHRNB2CHRNB4
SCHEMBL9030773 0.78 CHRNB2 (0.45) ACHEBDKRB1LTB4R2CHRNB2CHRNB4
SCHEMBL8958523 0.77 BDKRB1 (0.49) ACHEBDKRB1
SCHEMBL5782255 0.77 BDKRB1 (0.66) ACHEBDKRB1SLC6A3SLC6A4BRS3
SCHEMBL9030770 0.77 IDO1 (0.50) ACHEBDKRB1LTB4R2CHRNB2CHRNB4
SCHEMBL489306 0.76 NR1H2 (0.48) ACHELTB4R2SLC6A3SLC6A4BRS3
SCHEMBL8875151 0.76 ACHE (0.48) ACHELTB4R2SLC6A3SLC6A4BRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559233-A 3-/P-PHENYLBENZYL/IMIDAZOLONES AND PYRIMIDONES SANOFI (FR) 1996-09-24 US disclosed
US-5352788-A Angiotensin antagonist ELF SANOFI (FR) 1994-10-04 US disclosed
US-5270317-A N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present ELF SANOFI (FR) 1993-12-14 US disclosed