SCHEMBL8958291

SCHEMBL8958291

COC1=CC(=O)C(=O)C=C1N1CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HKDC1 Q2TB90 4/20 0.41
DNMT1 P26358 1/20 0.40
BCHE P06276 1/20 0.40
ACHE P22303 1/20 0.40
ERBB2 P04626 1/20 0.39
MAPT P10636 5/20 0.38
TP53 P04637 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HTT P42858 2/20 0.38
STAT3 P40763 1/20 0.38
IDO1 P14902 2/20 0.37
PTPN1 P18031 1/20 0.37
CDC25A P30304 1/20 0.37
CDC25B P30305 1/20 0.37
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CYP3A4 P08684 2/20 0.37
USP2 O75604 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8958544 0.77 DNMT1 (0.52) HKDC1DNMT1MAPTTP53SMN1; SMN2
SCHEMBL3417111 0.74 HKDC1 (0.56) HKDC1ERBB2MAPTTP53SMN1; SMN2
SCHEMBL1676679 0.71 DNMT1 (0.52) HKDC1DNMT1BCHEACHEMAPT
SCHEMBL8958416 0.71 MAPT (0.46) HKDC1DNMT1MAPTTP53SMN1; SMN2
SCHEMBL49737 0.69 ERBB2 (0.62) HKDC1ERBB2MAPTTP53SMN1; SMN2
SCHEMBL11025815 0.66 MAPT (0.50) HKDC1ERBB2MAPTTP53SMN1; SMN2
SCHEMBL9275509 0.64 HKDC1 (0.46) HKDC1ERBB2MAPTTP53SMN1; SMN2
SCHEMBL5485638 0.64 MAPT (0.61) HKDC1DNMT1MAPTTP53SMN1; SMN2
Triaziquone SCHEMBL7783197 0.62 MAPT (0.46) HKDC1DNMT1MAPTTP53SMN1; SMN2
Triaziquone SCHEMBL149876 0.62 MAPT (0.46) HKDC1DNMT1MAPTTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502214-A OXIDATION OF CATECHOL WITH OXIDANT, NUCLEOPHILIC REAGENT AND METAL CATALYST DANA FARBER CANCER INSTITUTE (US) 1996-03-26 US disclosed
WO-1995003267-A1 1,2-BENZOQUINONES DANA-FARBER CANCER INSTITUTE (US) 1995-02-02 WO disclosed