SCHEMBL8958804

SCHEMBL8958804

CC(=O)Nc1ccc(C(=O)C2CCN(CC(=O)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.72
LMNA P02545 2/20 0.72
HTT P42858 1/20 0.72
ALDH1A1 P00352 3/20 0.70
MEN1 O00255 2/20 0.64
KMT2A Q03164 2/20 0.64
POLB P06746 2/20 0.55
CYP2C19 P33261 3/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 2/20 0.54
CYP1A2 P05177 1/20 0.54
GAA P10253 1/20 0.54
UBE2N P61088 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
HTR7 P34969 1/20 0.53
HTR6 P50406 1/20 0.53
MAPT P10636 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
MAPK1 P28482 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9499649 0.88 SMN1; SMN2 (0.69) SMN1; SMN2LMNAHTTALDH1A1KMT2A
Hydrochloric Acid SCHEMBL9502312 0.86 SMN1; SMN2 (0.67) SMN1; SMN2LMNAHTTALDH1A1KMT2A
SCHEMBL9079271 0.85 KCNH2 (0.56) SMN1; SMN2LMNAHTTALDH1A1MEN1
SCHEMBL8958724 0.84 SMN1; SMN2 (0.63) SMN1; SMN2LMNAHTTALDH1A1MEN1
Hydrochloric Acid SCHEMBL9501099 0.82 LMNA (0.68) SMN1; SMN2LMNAHTTKMT2APOLB
SCHEMBL7302996 0.81 SMN1; SMN2 (0.59) SMN1; SMN2LMNAHTTALDH1A1MEN1
SCHEMBL27258181 0.81 SMN1; SMN2 (0.59) SMN1; SMN2LMNAHTTALDH1A1MEN1
SCHEMBL7302989 0.81 SMN1; SMN2 (0.59) SMN1; SMN2LMNAHTTALDH1A1MEN1
SCHEMBL6202951 0.81 LMNA (0.68) SMN1; SMN2LMNAHTTALDH1A1KMT2A
SCHEMBL27258188 0.81 SMN1; SMN2 (0.58) SMN1; SMN2LMNAHTTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500433-A PIPERIDINYL MEDICINAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-03-19 US disclosed
EP-0437790-B1 Antithrombotic compounds MERRELL DOW PHARMA (US) 1996-01-17 EP disclosed
US-5292752-A N-(p-fluorobenzoylmethyl)-4-(p-amidobenzoyl)piperidines MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0437790-A2 Antithrombotic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1991-07-24 EP disclosed