SCHEMBL8959024

SCHEMBL8959024

Fc1nc(OCc2ccccc2)c2[nH]cnc2n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 8/20 0.71
MGMT P16455 6/20 0.71
CDK1 P06493 3/20 0.71
CCNB1 P14635 3/20 0.71
CCNA2 P20248 3/20 0.71
CDK2 P24941 3/20 0.71
CCNA1 P78396 3/20 0.71
LMNA P02545 2/20 0.71
CYP1A2 P05177 1/20 0.71
CYP3A4 P08684 1/20 0.71
CYP2D6 P10635 1/20 0.71
CYP2C9 P11712 1/20 0.71
TSHR P16473 1/20 0.71
NFKB1 P19838 1/20 0.71
CYP2C19 P33261 1/20 0.71
BLM P54132 1/20 0.71
PMP22 Q01453 1/20 0.71
CDC7 O00311 3/20 0.63
DBF4 Q9UBU7 3/20 0.63
HTR2C P28335 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14542385 0.84 PIN1 (0.72) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL7437649 0.83 PIN1 (0.71) PIN1MGMTCDK1CCNB1CCNA2
6-O-Benzylguanine SCHEMBL61740 0.83 PIN1 (1.00) PIN1MGMTCDK1CCNB1CCNA2
6-O-Benzylguanine SCHEMBL31517079 0.83 PIN1 (1.00) PIN1MGMTCDK1CCNB1CCNA2
6-O-Benzylguanine SCHEMBL4631744 0.82 PIN1 (0.97) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL3303850 0.80 PIN1 (0.66) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL15759317 0.79 PIN1 (0.64) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL1404475 0.78 CDC7 (1.00) PIN1MGMTCDK1CCNB1CCNA2
6-O-Benzylguanine SCHEMBL4869639 0.78 PIN1 (0.88) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8959020 0.77 MGMT (0.46) PIN1MGMTCDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523100-B1 O6 -BENZYLATED GUANINE, GUANOSINE AND 2'-DEOXYGUANOSINE COMPOUNDS POSSESSING O6 -ALKYLGUANINE-DNA ALKYLTRANSFERASE DEPLETING ACTIVITY US HEALTH (US) 1996-08-28 EP disclosed
EP-0691981-A1 TUMOR TARGETING WITH L-ENANTIOMERIC OLIGONUCLEOTIDE CONJUGATES OF IMMUNOREAGENTS AND OF CHELATED RADIONUCLIDES THE WELLCOME FOUNDATION LIMITED (GB) 1996-01-17 EP disclosed
WO-1994020523-A1 TUMOR TARGETING WITH L-ENANTIOMERIC OLIGONUCLEOTIDE CONJUGATES OF IMMUNOREAGENTS AND OF CHELATED RADIONUCLIDES THE WELLCOME FOUNDATION LIMITED (GB) 1994-09-15 WO disclosed