SCHEMBL8959608

SCHEMBL8959608

C[C@@](N)(Cn1ccc2cc(F)c(F)cc21)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn1ccc2cc(F)c(F)cc21

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.45
HTR2C P28335 6/20 0.45
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HTR2B P41595 1/20 0.36
NPY5R Q15761 1/20 0.34
AR P10275 6/20 0.34
GRIN2B Q13224 1/20 0.33
KDM1A O60341 3/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27363223 0.91 HTR2A (0.49) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959713 0.91 HTR2A (0.49) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959561 0.91 HTR2A (0.49) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959864 0.91 HTR2A (0.49) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959551 0.90 AR (0.39) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959652 0.89 HTR2C (0.40) HTR2AHTR2CCYP1A2CYP3A4CYP2C9
SCHEMBL8959562 0.87 HTR2C (0.46) HTR2AHTR2CNPY5RARMTNR1A
SCHEMBL8959678 0.87 HTR2C (0.46) HTR2AHTR2CNPY5RARGRIN2B
SCHEMBL8959479 0.87 HTR2C (0.46) HTR2AHTR2CNPY5RARGRIN2B
SCHEMBL27356666 0.87 HTR2C (0.46) HTR2AHTR2CNPY5RARMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed