SCHEMBL8959678

SCHEMBL8959678

C[C@@](N)(Cn1ccc2cc(F)ccc21)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn1ccc2cc(F)ccc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.46
HTR2A P28223 2/20 0.46
AR P10275 5/20 0.43
FABP4 P15090 1/20 0.38
PPARG P37231 3/20 0.38
GRIN2B Q13224 1/20 0.35
NPY5R Q15761 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959479 1.00 HTR2C (0.46) HTR2CHTR2AARFABP4PPARG
SCHEMBL8959562 0.91 HTR2C (0.46) HTR2CHTR2AARFABP4PPARG
SCHEMBL27356666 0.91 HTR2C (0.46) HTR2CHTR2AARFABP4PPARG
SCHEMBL8959547 0.87 HTR2C (0.45) HTR2CHTR2AFABP4CDK4CCND1
SCHEMBL8959608 0.87 HTR2A (0.45) HTR2CHTR2AARGRIN2BNPY5R
SCHEMBL27342171 0.87 HTR2C (0.45) HTR2CHTR2AFABP4CDK4CCND1
SCHEMBL8959572 0.86 HTR2C (0.44) HTR2CHTR2AARFABP4PPARG
SCHEMBL8959588 0.86 HTR2A (0.46) HTR2CHTR2AARNPY5RCDK4
SCHEMBL27524962 0.86 HTR2A (0.46) HTR2CHTR2AARNPY5RCDK4
SCHEMBL27340857 0.86 HTR2A (0.46) HTR2CHTR2AARFABP4HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed