SCHEMBL8959643

SCHEMBL8959643

C[C@@](N)(Cn1ccc2c(C(F)(F)F)c(F)ccc21)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn1ccc2c(C(F)(F)F)c(F)ccc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.33
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
GRIN2B Q13224 2/20 0.31
NR3C1 P04150 2/20 0.30
PGR P06401 2/20 0.30
NR3C2 P08235 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959557 0.85 HTR2A (0.48) ARHTR2AHTR2CGRIN2BNR3C1
SCHEMBL8959753 0.85 HTR2A (0.48) ARHTR2AHTR2CGRIN2BNR3C1
SCHEMBL8959695 0.83 HTR2A (0.36) HTR2AHTR2CGRIN2B
SCHEMBL8959551 0.77 AR (0.39) ARHTR2AHTR2CGRIN2B
SCHEMBL8959608 0.77 HTR2A (0.45) ARHTR2AHTR2CGRIN2B
SCHEMBL8959711 0.77 HTR2C (0.45) ARHTR2AHTR2CNR3C1PGR
SCHEMBL8959479 0.76 HTR2C (0.46) ARHTR2AHTR2CGRIN2B
SCHEMBL8959678 0.76 HTR2C (0.46) ARHTR2AHTR2CGRIN2B
SCHEMBL8959588 0.74 HTR2A (0.46) ARHTR2AHTR2C
SCHEMBL27524962 0.74 HTR2A (0.46) ARHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed