SCHEMBL8959588

SCHEMBL8959588

C[C@@](N)(Cn1ccc2cc(Cl)ccc21)OC(=O)/C=C/C(=O)O[C@](C)(N)Cn1ccc2cc(Cl)ccc21

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
KRAS P01116 2/20 0.42
ACLY P53396 2/20 0.38
OXER1 Q8TDS5 1/20 0.38
KMO O15229 1/20 0.37
P2RX3 P56373 4/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NPY5R Q15761 1/20 0.35
AR P10275 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CCR2 P41597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27524962 1.00 HTR2A (0.46) HTR2AHTR2CKRASACLYOXER1
SCHEMBL7997832 0.91 KMO (0.48) HTR2AHTR2CACLYOXER1KMO
SCHEMBL27342171 0.87 HTR2C (0.45) HTR2AHTR2CHDAC3HDAC1HDAC2
SCHEMBL8959547 0.87 HTR2C (0.45) HTR2AHTR2CHDAC3HDAC1HDAC2
SCHEMBL8959678 0.86 HTR2C (0.46) HTR2AHTR2CHDAC3HDAC1HDAC2
SCHEMBL27340857 0.86 HTR2A (0.46) HTR2AHTR2CKRASHDAC3HDAC1
SCHEMBL8959479 0.86 HTR2C (0.46) HTR2AHTR2CHDAC3HDAC1HDAC2
SCHEMBL8959618 0.86 HTR2A (0.46) HTR2AHTR2CKRASHDAC3HDAC1
SCHEMBL8959561 0.83 HTR2A (0.49) HTR2AHTR2CKRASKMOHDAC1
SCHEMBL8959864 0.83 HTR2A (0.49) HTR2AHTR2CKRASKMOHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed