SCHEMBL8959872

SCHEMBL8959872

CC(=O)Oc1cn(C(C)=O)c2ccc(F)c(Cl)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
NOTUM Q6P988 2/20 0.36
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
EP300 Q09472 1/20 0.31
CREBBP Q92793 1/20 0.31
KDM4E B2RXH2 3/20 0.30
TDP1 Q9NUW8 2/20 0.30
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
ALDH1A1 P00352 1/20 0.30
ESR1 P03372 1/20 0.30
ITGB3 P05106 1/20 0.30
ITGA2B P08514 1/20 0.30
HMGB1 P09429 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
GGT1 P19440 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959947 0.87 NOTUM (0.37) NOTUMMEN1KMT2AKDM4ENPC1
SCHEMBL32691742 0.83 NOTUM (0.36) NOTUMKDM4ETDP1NPC1RAB9A
SCHEMBL3564119 0.81 NOTUM (0.41) NOTUMMEN1KMT2AEP300CREBBP
SCHEMBL28977332 0.80 CYP4F2 (0.37) CYP4F2CYP4A11NOTUMKMT2AEP300
SCHEMBL28977327 0.77 NOTUM (0.48) NOTUMMEN1KMT2AKDM4ETDP1
SCHEMBL27363222 0.76 NOTUM (0.37) NOTUMMEN1KMT2AEP300CREBBP
SCHEMBL2476989 0.74 ABCB11 (0.46) NOTUMMEN1KMT2AKDM4ETDP1
SCHEMBL28977329 0.71 EGFR (0.37) NOTUMKMT2AKDM4ETDP1NPC1
SCHEMBL3241798 0.71 ABCB11 (0.46) NOTUMMEN1KMT2ACREBBPKDM4E
SCHEMBL8959923 0.71 KDM4E (0.37) CYP4F2CYP4A11NOTUMCREBBPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
CN-1105988-A 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed