SCHEMBL8960256

SCHEMBL8960256

CC(C)(C)c1ccccc1C#C[Si](C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
TSHR P16473 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.39
CA2 P00918 1/20 0.35
CREBBP Q92793 1/20 0.33
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
KIF11 P52732 1/20 0.31
GRIN2D O15399 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347622 0.82 FFAR1 (0.40) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL3839029 0.80 KDM4E (0.49) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL17940722 0.77 KDM4E (0.36) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL26259528 0.74 ALDH1A1 (0.32) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL10535351 0.74 TSHR (0.45) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL563737 0.73 NPC1 (0.50) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL26259658 0.73 KDM4E (0.31) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL31349196 0.72 TSHR (0.48) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL1324387 0.72 TSHR (0.48) ALDH1A1TSHRKDM4EMEN1CYP1A2
SCHEMBL26259915 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516904-A SKIN AND IMMUNE DISORDERS; ANTIARTHRITIC AGENTS; WOUND HEALING AGENTS ALLERGAN, INC. (US) 1996-05-14 US disclosed
EP-0436398-B1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN INC (US) 1996-01-31 EP disclosed
US-5414007-A Skin disorders ALLERGAN, INC. (US) 1995-05-09 US disclosed
US-5349105-A Skin disorder ALLERGAN, INC. (US) 1994-09-20 US disclosed
US-5264456-A Skin disorders, anticarcinogenic agents, antiarthritic agents, immunology or wound healing agents ALLERGAN, INC. (US) 1993-11-23 US disclosed
US-5202471-A Skin disorders ALLERGAN, INC. (US) 1993-04-13 US disclosed
US-5175185-A Antiacne agents ALLERGAN, INC. (US) 1992-12-29 US disclosed
EP-0436398-A1 Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity ALLERGAN, INC. (US) 1991-07-10 EP disclosed
US-5013744-A Skin disorders ALLERGAN, INC. (US) 1991-05-07 US disclosed