SCHEMBL8961789

SCHEMBL8961789

CN(C)CC(=O)c1cc2c(cc1N)OCO2

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 6/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
GAA P10253 2/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.41
LMNA P02545 1/20 0.41
L3MBTL4 Q8NA19 1/20 0.39
HPGD P15428 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
POLB P06746 1/20 0.38
MCL1 Q07820 1/20 0.38
HSD17B10 Q99714 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980406 0.79 NPC1 (0.48) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL8041232 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL21450331 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL29084683 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL30884756 0.79 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL8961778 0.77 KDM4E (0.55) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL30014749 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL209949 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL24642665 0.76 KDM4E (0.47) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL25333842 0.75 KDM4E (0.42) ALDH1A1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559235-A ANTITUMOR GLAXO WELLCOME INC. (US) 1996-09-24 US disclosed
EP-0540099-B1 Water soluble camptothecin derivatives GLAXO WELLCOME INC (US) 1996-04-17 EP disclosed
US-5342947-A Treating alkylenedioxy-7-trihaloacetamidomethylenecamptothecin with hydrochloric or sulfuric acid to yield amine salt, treating with alkali metal hydroxide or carbonate to obtain free base GLAXO INC. (US) 1994-08-30 US disclosed
EP-0540099-A1 Water soluble camptothecin derivatives GLAXO WELLCOME INC. (US) 1993-05-05 EP disclosed