SCHEMBL8961878

SCHEMBL8961878

CC/C=C/COC(=O)CC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
NAAA Q02083 1/20 0.40
NR1I2 O75469 1/20 0.40
PGR P06401 1/20 0.40
PTGS2 P35354 1/20 0.40
PDE4D Q08499 1/20 0.40
ALDH1A1 P00352 6/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 2/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
BLM P54132 1/20 0.36
WRN Q14191 1/20 0.36
HIF1A Q16665 1/20 0.36
OXER1 Q8TDS5 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11292223 0.93 NAAA (0.44) NAAAALDH1A1TSHRALOX15HSD17B10
SCHEMBL8744195 0.93 NAAA (0.44) NAAAALDH1A1TSHRALOX15HSD17B10
SCHEMBL8744192 0.93 NAAA (0.44) NAAAALDH1A1TSHRALOX15HSD17B10
SCHEMBL30902248 0.84 ALDH1A1 (0.44) NAAAPGRALDH1A1TSHRALOX15
SCHEMBL30902264 0.84 ALDH1A1 (0.44) NAAAPGRALDH1A1TSHRALOX15
SCHEMBL2039597 0.82 NAAA (0.42) PTGS1ADORA3NAAANR1I2PGR
SCHEMBL17391650 0.82 TSHR (0.41) PTGS1ADORA3NR1I2PGRPTGS2
SCHEMBL873463 0.82 NAAA (0.42) PTGS1ADORA3NAAANR1I2PGR
SCHEMBL21467458 0.82 NAAA (0.38) NAAAALDH1A1TSHRALOX15CYP1A2
SCHEMBL873462 0.82 NAAA (0.42) PTGS1ADORA3NAAANR1I2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523543-B1 Chiral piperazine derivatives HOFFMANN LA ROCHE (CH) 1996-02-07 EP disclosed
US-5356559-A Optically active piperazinyl derivatives as liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-10-18 US disclosed
EP-0523543-A1 Chiral piperazine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-01-20 EP disclosed