SCHEMBL8962813

SCHEMBL8962813

Fc1cc([C@H]2CC[C@H](/C=C/Cl)CC2)ccc1Br

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.44
KCNH2 Q12809 2/20 0.44
KDM1B Q8NB78 1/20 0.44
RCOR1 Q9UKL0 1/20 0.37
HDAC2 Q92769 1/20 0.35
IDO1 P14902 1/20 0.31
EP300 Q09472 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962804 1.00 KDM1A (0.44) KDM1AKCNH2KDM1BRCOR1HDAC2
SCHEMBL8962935 0.96 KDM1A (0.41) KDM1AKCNH2KDM1BRCOR1HDAC2
SCHEMBL8962923 0.89 KDM1A (0.37) KDM1AKCNH2KDM1BRCOR1HDAC2
SCHEMBL8962932 0.89 KDM1A (0.37) KDM1AKCNH2KDM1BRCOR1HDAC2
SCHEMBL8962808 0.86 KDM1A (0.36) KDM1AKCNH2HDAC2
SCHEMBL8962817 0.86 KDM1A (0.36) KDM1AKCNH2HDAC2
SCHEMBL17780006 0.83 KDM1A (0.58) KDM1AKCNH2KDM1BRCOR1IDO1
SCHEMBL8962613 0.83 SLC6A2 (0.35) KCNH2HDAC2
SCHEMBL8962617 0.83 SLC6A2 (0.35) KCNH2HDAC2
SCHEMBL8963266 0.82 SLC6A3 (0.35) HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed