SCHEMBL8963128

SCHEMBL8963128

CCOc1ccc(-c2cnc([C@H]3CC[C@H](/C=C/Cl)CC3)nc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.38
MAPT P10636 5/20 0.38
KDM4E B2RXH2 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.36
TP53 P04637 1/20 0.36
NQO1 P15559 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
GRM2 Q14416 1/20 0.34
CHRNA7 P36544 2/20 0.34
TNK2 Q07912 1/20 0.34
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
NLRP3 Q96P20 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300329 0.90 ACACB (0.39) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL8962894 0.87 KDR (0.36) NPC1RAB9AMEN1KMT2ACASP3
SCHEMBL8962664 0.86 HDAC1 (0.32) NQO1KMT2ACACNA2D1
SCHEMBL8962673 0.86 HDAC1 (0.32) NQO1KMT2ACACNA2D1
SCHEMBL8962700 0.85 NQO1 (0.39) XDHMAPTKDM4ENPC1RAB9A
SCHEMBL8962695 0.85 NQO1 (0.39) XDHMAPTKDM4ENPC1RAB9A
SCHEMBL8962929 0.84 EP300 (0.34) NPC1RAB9ATP53
SCHEMBL8962996 0.82 LRRK2 (0.36) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL8962887 0.82 NISCH (0.33) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL9300971 0.81 MAP4K1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed