SCHEMBL9300971

SCHEMBL9300971

COCc1ccc(-c2cnc([C@H]3CC[C@H](/C=C/Cl)CC3)nc2)cc1

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.32
NAAA Q02083 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
HDAC5 Q9UQL6 2/20 0.31
GPR88 Q9GZN0 1/20 0.31
ERN1 O75460 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
HDAC4 P56524 1/20 0.31
PDE10A Q9Y233 1/20 0.31
HTR6 P50406 1/20 0.30
PTGS2 P35354 1/20 0.30
PTGES O14684 1/20 0.30
CHRM1 P11229 2/20 0.30
GPR119 Q8TDV5 1/20 0.30
SYK P43405 1/20 0.30
FEN1 P39748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962769 0.87 PDE10A (0.32) PDE10A
SCHEMBL8962773 0.87 PDE10A (0.32) PDE10A
SCHEMBL8962929 0.86 EP300 (0.34) HDAC4PDE10A
SCHEMBL8962953 0.84 HDAC2 (0.35) ERN1HTR6PTGS2
SCHEMBL8962947 0.84 HDAC2 (0.35) ERN1HTR6PTGS2
SCHEMBL8962887 0.84 NISCH (0.33) FFAR4GPR88HDAC4
SCHEMBL8962894 0.83 KDR (0.36) PTGS2
SCHEMBL8963259 0.81 RARB (0.36) FFAR4
SCHEMBL8962996 0.81 LRRK2 (0.36) HDAC4
SCHEMBL8963128 0.81 XDH (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed