SCHEMBL8962929

SCHEMBL8962929

CCc1ccc(-c2cnc([C@H]3CC[C@H](/C=C/Cl)CC3)nc2)cc1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
S1PR1 P21453 1/20 0.33
S1PR5 Q9H228 1/20 0.33
HDAC4 P56524 1/20 0.32
TP53 P04637 2/20 0.32
METAP2 P50579 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30
KDM1A O60341 1/20 0.30
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962887 0.90 NISCH (0.33) NPC1RAB9AS1PR1S1PR5HDAC4
SCHEMBL8963259 0.87 RARB (0.36) NPC1GAARAB9AS1PR1S1PR5
SCHEMBL8962857 0.86 SPHK1 (0.40) NPC1GAARAB9A
SCHEMBL9300971 0.86 MAP4K1 (0.32) HDAC4PDE10A
SCHEMBL8962927 0.86 PDE8B (0.31) PDE10A
SCHEMBL8962934 0.86 PDE8B (0.31) PDE10A
SCHEMBL8962996 0.85 LRRK2 (0.36) NPC1RAB9AHDAC4TP53EGLN1
SCHEMBL8963128 0.84 XDH (0.38) NPC1RAB9ATP53
SCHEMBL8962835 0.83 SPHK1 (0.36) EP300NPC1RAB9AS1PR1S1PR5
SCHEMBL8962826 0.83 SPHK1 (0.36) EP300NPC1RAB9AS1PR1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed