SCHEMBL8962996

SCHEMBL8962996

Cc1ccc(-c2cnc([C@H]3CC[C@H](/C=C/Cl)CC3)nc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 2/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC4 P56524 1/20 0.34
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
TP53 P04637 1/20 0.32
HTT P42858 1/20 0.32
EGLN1 Q9GZT9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962929 0.85 EP300 (0.34) NPC1RAB9AHDAC4TP53EGLN1
SCHEMBL8962894 0.85 KDR (0.36) NPC1RAB9AHTR2AHTR2CHTR2B
SCHEMBL8963386 0.84 PDE10A (0.33)
SCHEMBL8963391 0.84 PDE10A (0.33)
SCHEMBL8962887 0.82 NISCH (0.33) NPC1RAB9ASMN1; SMN2MAPTHDAC4
SCHEMBL8963128 0.82 XDH (0.38) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL8962852 0.81 SLC18A3 (0.39) LRRK2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL8962862 0.81 SLC18A3 (0.39) LRRK2NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL9300971 0.81 MAP4K1 (0.32) HDAC4
SCHEMBL9300329 0.80 ACACB (0.39) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed