SCHEMBL8963223

SCHEMBL8963223

Fc1cc([C@H]2CC[C@H](/C=C/Cl)CC2)ccc1OC(F)F

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.35
PDE10A Q9Y233 1/20 0.35
MGLL Q99685 2/20 0.33
KDM1A O60341 2/20 0.31
TLR9 Q9NR96 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963217 1.00 PDE2A (0.35) PDE2APDE10AMGLLKDM1ATLR9
SCHEMBL8962853 0.96 PDE2A (0.36) PDE2APDE10AMGLL
SCHEMBL8963112 0.90 JAK2 (0.34) PDE2APDE10A
SCHEMBL8963104 0.90 JAK2 (0.34) PDE2APDE10A
SCHEMBL8454674 0.82 MGLL (0.33) PDE2APDE10AMGLL
SCHEMBL8454678 0.82 MGLL (0.33) PDE2APDE10AMGLL
SCHEMBL8963018 0.82 EPHX2 (0.36) PDE2AKDM1A
SCHEMBL8963026 0.82 EPHX2 (0.36) PDE2AKDM1A
SCHEMBL8963152 0.81 PDE2A (0.31) PDE2APDE10A
SCHEMBL8448650 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed