SCHEMBL8963733

SCHEMBL8963733

Cc1[nH]c(-c2ccccc2)nc1C(=O)C(C(c1ccccc1)c1ccccc1)N1CCNCC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 8/20 0.51
SLC9A1 P19634 1/20 0.42
OPRD1 P41143 7/20 0.40
PRMT5 O14744 1/20 0.39
MAPT P10636 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963679 0.76 MEN1 (0.42) PIN1OPRD1PRMT5MEN1KMT2A
Hydrochloric Acid SCHEMBL8963658 0.75 MEN1 (0.39) PIN1OPRD1PRMT5MAPTMEN1
SCHEMBL8964151 0.73 PIN1 (0.71) PIN1SLC9A1MAPTCYP1A2MAPK1
SCHEMBL8963580 0.71 PRMT5 (0.40) OPRD1PRMT5MEN1KMT2ACYP1A2
Hydrochloric Acid SCHEMBL8963783 0.70 PRMT5 (0.40) OPRD1PRMT5MEN1KMT2ACYP1A2
Hydrochloric Acid SCHEMBL8963905 0.70 PIN1 (0.36) PIN1OPRD1PRMT5MAPTMEN1
SCHEMBL11564100 0.70 PIN1 (0.81) PIN1SLC9A1MAPTCYP1A2MAPK1
SCHEMBL316552 0.70 PIN1 (1.00) PIN1SLC9A1MAPTCYP1A2MAPK1
SCHEMBL8963723 0.70 PIN1 (0.51) PIN1SLC9A1MEN1KMT2A
SCHEMBL8963650 0.70 CHEK2 (0.40) OPRD1PRMT5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed