SCHEMBL8963977

SCHEMBL8963977

Cc1ccc(-c2nc(N3CCN(C(c4ccccc4C(C)(C)C)c4ccccc4C(C)(C)C)CC3)c(C)[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 2/20 0.35
DGAT1 O75907 2/20 0.33
MAPT P10636 2/20 0.33
ACHE P22303 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
RBP4 P02753 1/20 0.33
MAOB P27338 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HSD17B10 Q99714 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963517 0.82 DRD2 (0.49) DRD2DRD4DRD3GNRHRCYP3A4
Hydrochloric Acid SCHEMBL8963906 0.77 PIN1 (0.34) NPY5RMAPTDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL8964006 0.75 DRD2 (0.34) NPY5RMAPTDRD2DRD4DRD3
SCHEMBL8963527 0.72 PRMT5 (0.32) DRD2DRD4DRD3TRPV1TNKS
Hydrochloric Acid SCHEMBL8964045 0.72 MEN1 (0.39) MAPTDRD2DRD4DRD3
SCHEMBL8963694 0.69 TRPV1 (0.37) TRPV1GNRHR
SCHEMBL8963847 0.69 DRD2 (0.53) DRD2DRD4DRD3CYP3A4CYP2C9
SCHEMBL8963984 0.67 DRD2 (0.51) DRD2DRD4DRD3CYP3A4CYP2C9
SCHEMBL8963495 0.67 DRD2 (0.50) MAPTDRD2DRD4DRD3ALDH1A1
SCHEMBL8963742 0.67 MEN1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514800-A CALCIUM CHANNEL BLOCKERS, CEREBRAL ISCHEMIA SYNTEX PHARMACEUTICALS, LTD. (GB) 1996-05-07 US disclosed