SCHEMBL8964976

SCHEMBL8964976

N#C[C@@H](OC(=O)Cc1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.56
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
PAM P19021 1/20 0.45
KLK7 P49862 3/20 0.44
CNR2 P34972 1/20 0.42
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
AKR1B1 P15121 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CNR1 P21554 1/20 0.40
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11025357 1.00 TSHR (0.56) TSHRALDH1A1MAPK1L3MBTL1CRHBP
SCHEMBL8964825 0.87 KLK7 (0.59) TSHRALDH1A1L3MBTL1KLK7CNR2
SCHEMBL10780199 0.85 TSHR (0.57) TSHRALDH1A1MAPK1L3MBTL1CRHBP
SCHEMBL8965076 0.85 ALDH1A1 (0.51) TSHRALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL1200602 0.84 TSHR (0.45) TSHRALDH1A1MAPK1L3MBTL1CRHBP
SCHEMBL27836917 0.82 TSHR (0.40) TSHRALDH1A1SMN1; SMN2KDM4ELMNA
SCHEMBL8965109 0.81 TSHR (0.49) TSHRALDH1A1MAPK1L3MBTL1PAM
SCHEMBL8965028 0.79 TSHR (0.46) TSHRALDH1A1L3MBTL1SMN1; SMN2LMNA
SCHEMBL10992713 0.79 ALDH1A1 (0.43) TSHRALDH1A1
SCHEMBL18671086 0.79 TSHR (0.67) TSHRALDH1A1MAPK1L3MBTL1PAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493047-A REACTING OPTICALLY ACTIVE CYANOHYDRIN WITH CARBOXYLIC ACID IN PRESENCE OF DIALKYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE TO FORM ESTER OF OPPOSITE CONFIGURATION DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1996-02-20 US disclosed
EP-0601237-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed
EP-0601632-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed