SCHEMBL8965028

SCHEMBL8965028

COCC(=O)O[C@H](C#N)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
GAA P10253 1/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 4/20 0.38
TDP1 Q9NUW8 2/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C1 Q04828 1/20 0.37
HPGD P15428 1/20 0.37
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
USP2 O75604 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.36
CA12 O43570 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27836917 0.84 TSHR (0.40) TSHRGAAKMT2AALDH1A1TDP1
SCHEMBL10992713 0.81 ALDH1A1 (0.43) TSHRKMT2AALDH1A1TDP1MEN1
SCHEMBL8964976 0.79 TSHR (0.56) TSHRALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL11025357 0.79 TSHR (0.56) TSHRALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL7699172 0.78 ALDH1A1 (0.50) TSHRKMT2AALDH1A1TDP1MAPT
SCHEMBL3071211 0.78 TSHR (0.53) TSHRKMT2AALDH1A1MAPTMEN1
SCHEMBL2835326 0.78 ALDH1A1 (0.50) TSHRKMT2AALDH1A1TDP1MAPT
SCHEMBL8964825 0.77 KLK7 (0.59) TSHRALDH1A1TDP1SMN1; SMN2USP2
SCHEMBL1766133 0.77 TSHR (0.51) TSHRKMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL5932426 0.76 TSHR (0.45) TSHRKMT2AALDH1A1TDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493047-A REACTING OPTICALLY ACTIVE CYANOHYDRIN WITH CARBOXYLIC ACID IN PRESENCE OF DIALKYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE TO FORM ESTER OF OPPOSITE CONFIGURATION DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1996-02-20 US disclosed
EP-0601237-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed
EP-0601632-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed