SCHEMBL8965076

SCHEMBL8965076

N#C[C@@H](OC(=O)Cc1ccc([N+](=O)[O-])cc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
MAPT P10636 3/20 0.50
HTT P42858 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
OPRK1 P41145 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
GAA P10253 2/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11025357 0.85 TSHR (0.56) ALDH1A1L3MBTL1SMN1; SMN2TSHR
SCHEMBL8964976 0.85 TSHR (0.56) ALDH1A1L3MBTL1SMN1; SMN2TSHR
SCHEMBL6676165 0.83 ALDH1A1 (0.56) ALDH1A1MAPTHTTNPSR1OPRM1
SCHEMBL8965070 0.81 CES1 (0.49) ALDH1A1MAPTNPSR1OPRK1MEN1
SCHEMBL8964825 0.80 KLK7 (0.59) ALDH1A1L3MBTL1SMN1; SMN2TDP1TSHR
SCHEMBL7262891 0.78 CES2 (0.49) ALDH1A1MAPTNPSR1CYP2C19OPRK1
SCHEMBL8964999 0.75 LMNA (0.45) ALDH1A1MAPTHTTCYP1A2CYP2C19
SCHEMBL27836917 0.72 TSHR (0.40) ALDH1A1MEN1KMT2AGAASMN1; SMN2
SCHEMBL10780199 0.72 TSHR (0.57) ALDH1A1L3MBTL1SMN1; SMN2TSHR
SCHEMBL1200602 0.72 TSHR (0.45) ALDH1A1L3MBTL1SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493047-A REACTING OPTICALLY ACTIVE CYANOHYDRIN WITH CARBOXYLIC ACID IN PRESENCE OF DIALKYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE TO FORM ESTER OF OPPOSITE CONFIGURATION DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1996-02-20 US disclosed
EP-0601237-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed
EP-0601632-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed