SCHEMBL8965070

SCHEMBL8965070

N#C[C@@H](OC(=O)c1ccc([N+](=O)[O-])cc1)c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.49
CES2 O00748 1/20 0.49
KMT2A Q03164 5/20 0.46
MEN1 O00255 4/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 3/20 0.46
ALOX5 P09917 1/20 0.46
MAPK1 P28482 2/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 2/20 0.45
CYP1B1 Q16678 1/20 0.45
HSP90AA1 P07900 1/20 0.45
OPRK1 P41145 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
SRD5A2 P31213 1/20 0.42
BCHE P06276 1/20 0.42
MAOB P27338 1/20 0.42
CRHBP P24387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7262891 0.95 CES2 (0.49) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL2453510 0.84 TSHR (0.52) KMT2AMEN1ALDH1A1MAPTPOLB
SCHEMBL8964823 0.84 TSHR (0.52) KMT2AMEN1ALDH1A1MAPTPOLB
SCHEMBL8965076 0.81 ALDH1A1 (0.51) KMT2AMEN1ALDH1A1MAPTTDP1
SCHEMBL1142464 0.79 CES1 (0.53) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL8964973 0.78 MAPT (0.60) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL14662793 0.77 MEN1 (0.63) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL19926029 0.76 CES1 (0.53) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL16398922 0.75 KMT2A (0.57) CES1CES2KMT2AMEN1ALDH1A1
SCHEMBL7239333 0.74 TP53 (0.45) KMT2AMEN1ALDH1A1POLBESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5493047-A REACTING OPTICALLY ACTIVE CYANOHYDRIN WITH CARBOXYLIC ACID IN PRESENCE OF DIALKYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE TO FORM ESTER OF OPPOSITE CONFIGURATION DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1996-02-20 US disclosed
EP-0601237-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed
EP-0601632-A1 Method of preparing optically active cyanohydrin derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1994-06-15 EP disclosed