SCHEMBL8965199

SCHEMBL8965199

C[C@@H](/C=C/c1cccc(-c2cccc(F)c2)c1)NO

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 8/20 0.46
RELA Q04206 4/20 0.42
PTGS1 P23219 3/20 0.41
PTGS2 P35354 1/20 0.41
ESR2 Q92731 1/20 0.41
NQO2 P16083 1/20 0.41
KDM1A O60341 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
MMP13 P45452 1/20 0.40
MMP14 P50281 1/20 0.40
FBP1 P09467 1/20 0.40
TRPM2 O94759 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965132 0.90 BCL2L1 (0.48) NFE2L2RELAPTGS2ESR2KDM1A
SCHEMBL8965558 0.90 BCL2L1 (0.48) NFE2L2RELAPTGS2ESR2KDM1A
SCHEMBL8965561 0.90 BCL2L1 (0.48) NFE2L2RELAPTGS2ESR2KDM1A
SCHEMBL9063419 0.81 HDAC2 (0.43) RELAPTGS2MMP1MMP2MMP3
SCHEMBL9063905 0.81 HDAC2 (0.43) RELAPTGS2MMP1MMP2MMP3
SCHEMBL8965195 0.78 RELA (0.49) NFE2L2RELANQO2HDAC1HDAC6
SCHEMBL8964911 0.78 CYP17A1 (0.48) NFE2L2RELAPTGS1PTGS2NQO2
SCHEMBL8964908 0.78 CYP17A1 (0.48) NFE2L2RELAPTGS1PTGS2NQO2
SCHEMBL8964910 0.78 CYP17A1 (0.48) NFE2L2RELAPTGS1PTGS2NQO2
SCHEMBL8964905 0.78 CYP17A1 (0.48) NFE2L2RELAPTGS1PTGS2NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696271-A1 CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITING HYDROXAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025430-A1 CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITING HYDROXAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1994-11-10 WO disclosed