SCHEMBL8966468

SCHEMBL8966468

O=C(N(CCSc1ccncc1)Cc1ccccc1)C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 5/20 0.44
CYP2C9 P11712 4/20 0.44
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2D6 P10635 2/20 0.44
HIF1A Q16665 1/20 0.44
ALDH1A1 P00352 3/20 0.39
CES1 P23141 1/20 0.39
LMNA P02545 3/20 0.39
KMT2A Q03164 4/20 0.38
HTT P42858 3/20 0.38
MEN1 O00255 3/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
MAPT P10636 1/20 0.37
CHRM1 P11229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966758 0.93 CYP2C19 (0.43) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8966480 0.92 CYP2C19 (0.42) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL8966760 0.83 CYP1A2 (0.48) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL8621464 0.81 ALDH1A1 (0.50) CYP1A2CYP3A4ALDH1A1LMNAKMT2A
SCHEMBL8966793 0.78 HDAC1 (0.37) CYP1A2ALDH1A1KMT2AMEN1SMN1; SMN2
Hydrochloric Acid SCHEMBL8966715 0.77 L3MBTL1 (0.38) ALDH1A1LMNAKMT2AMEN1SMN1; SMN2
SCHEMBL9252468 0.77 CYP1A2 (0.43) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL8967239 0.76 LPAR1 (0.46) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL8966322 0.76 CYP2C9 (0.46) CYP2C19CYP2C9CYP1A2CYP3A4CYP2D6
SCHEMBL16373478 0.76 CES1 (0.52) CYP2C19CYP2C9CYP1A2ALDH1A1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
EP-0522606-B1 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-04-03 EP disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed