SCHEMBL8966730

SCHEMBL8966730

CC(=O)N(CCCSc1ccncc1)Cc1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
CYP1A2 P05177 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.40
HDAC1 Q13547 2/20 0.39
MAPT P10636 1/20 0.39
LIN28A Q9H9Z2 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
HSP90AA1 P07900 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8966687 0.99 ALDH1A1 (0.41) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
SCHEMBL8967342 0.86 HDAC1 (0.44) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
SCHEMBL8616106 0.85 ALDH1A1 (0.48) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
Hydrochloric Acid SCHEMBL8966843 0.85 L3MBTL1 (0.46) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
SCHEMBL8966793 0.85 HDAC1 (0.37) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
Hydrochloric Acid SCHEMBL8617887 0.84 ALDH1A1 (0.47) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1
Hydrochloric Acid SCHEMBL8966715 0.84 L3MBTL1 (0.38) ALDH1A1SMN1; SMN2HDAC1MAPTLIN28A
SCHEMBL8966322 0.84 CYP2C9 (0.46) ALDH1A1CYP1A2TSHRMAPTMEN1
Hydrochloric Acid SCHEMBL8967045 0.83 CYP2C9 (0.44) ALDH1A1CYP1A2TSHRMAPTMEN1
SCHEMBL2189143 0.78 TRPM8 (0.47) ALDH1A1CYP1A2TSHRSMN1; SMN2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed