SCHEMBL8967729

SCHEMBL8967729

O=C(CCCN1CC[C@](O)(c2ccccc2)[C@@H](C(O)c2ccccc2)C1)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
TSHR P16473 1/20 0.63
DRD2 P14416 3/20 0.58
LMNA P02545 2/20 0.52
KMT2A Q03164 2/20 0.52
DRD3 P35462 2/20 0.48
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967685 0.94 ALDH1A1 (0.65) ALDH1A1TSHRDRD2LMNAKMT2A
SCHEMBL8966878 0.93 DRD2 (0.62) ALDH1A1TSHRDRD2KMT2ADRD3
SCHEMBL9181467 0.93 ALDH1A1 (0.58) ALDH1A1TSHRDRD2LMNAKMT2A
SCHEMBL8967606 0.91 DRD2 (0.57) ALDH1A1TSHRDRD2KMT2ADRD3
SCHEMBL9711034 0.87 ALDH1A1 (0.68) ALDH1A1TSHRDRD2LMNAKMT2A
SCHEMBL8967661 0.86 DRD2 (0.60) TSHRDRD2KMT2ADRD3MEN1
SCHEMBL8967611 0.86 DRD2 (0.60) TSHRDRD2KMT2ADRD3MEN1
SCHEMBL9173912 0.85 ALDH1A1 (0.71) ALDH1A1TSHRDRD2LMNAKMT2A
SCHEMBL11861506 0.83 ALDH1A1 (0.68) ALDH1A1TSHRLMNAKMT2ASLC6A3
SCHEMBL11867863 0.83 ALDH1A1 (0.68) ALDH1A1TSHRLMNAKMT2ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512584-A 1,3,4-trisubstituted piperidine derivatives, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1996-04-30 US disclosed
EP-0580644-B1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE BASF AG (DE) 1995-06-28 EP disclosed
WO-1992018480-A1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1992-10-29 WO disclosed