SCHEMBL8967606

SCHEMBL8967606

O=C(CCCN1CC[C@](O)(c2ccc(F)cc2)[C@@H](C(O)c2ccc(F)cc2)C1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.57
CYP2D6 P10635 3/20 0.54
TSHR P16473 2/20 0.53
ALDH1A1 P00352 1/20 0.53
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
HTR1A P08908 2/20 0.50
ADRA2A P08913 2/20 0.50
CHRM1 P11229 2/20 0.50
ADRA2B P18089 2/20 0.50
ADRA2C P18825 2/20 0.50
CHRM3 P20309 2/20 0.50
SLC6A2 P23975 2/20 0.50
HTR2A P28223 2/20 0.50
SLC6A4 P31645 2/20 0.50
ADRA1A P35348 2/20 0.50
HRH1 P35367 2/20 0.50
OPRM1 P35372 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967611 0.95 DRD2 (0.60) DRD2CYP2D6TSHRMEN1KMT2A
SCHEMBL8967661 0.95 DRD2 (0.60) DRD2CYP2D6TSHRMEN1KMT2A
SCHEMBL8966878 0.94 DRD2 (0.62) DRD2CYP2D6TSHRALDH1A1MEN1
SCHEMBL8967729 0.91 ALDH1A1 (0.63) DRD2CYP2D6TSHRALDH1A1MEN1
SCHEMBL8967685 0.85 ALDH1A1 (0.65) DRD2TSHRALDH1A1MEN1KMT2A
SCHEMBL9181467 0.85 ALDH1A1 (0.58) DRD2CYP2D6TSHRALDH1A1KMT2A
SCHEMBL8967036 0.83 ALDH1A1 (0.63) DRD2TSHRALDH1A1HTR1AHTR2A
SCHEMBL8967710 0.82 KMT2A (0.66) DRD2CYP2D6TSHRALDH1A1MEN1
SCHEMBL9711021 0.80 ALDH1A1 (0.64) DRD2TSHRALDH1A1MEN1KMT2A
SCHEMBL8966947 0.80 KMT2A (0.69) DRD2ALDH1A1MEN1KMT2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512584-A 1,3,4-trisubstituted piperidine derivatives, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1996-04-30 US disclosed