SCHEMBL8968849

SCHEMBL8968849

N#Cc1ccc(-c2ccccc2)c(NC(=O)Nc2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
CXCR1 P25024 1/20 0.53
CXCR2 P25025 1/20 0.53
HTT P42858 2/20 0.51
MET P08581 1/20 0.50
KDR P35968 1/20 0.50
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
MAPT P10636 4/20 0.49
LMNA P02545 3/20 0.49
ATM Q13315 1/20 0.49
GRIK1 P39086 1/20 0.48
AHR P35869 1/20 0.48
IDH2 P48735 1/20 0.48
KDM4E B2RXH2 2/20 0.47
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPK1 P28482 1/20 0.46
NPC1 O15118 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8969388 0.81 HSD17B10 (0.53) CYP11B1CYP11B2CXCR1CXCR2HTT
SCHEMBL8968218 0.81 CYP11B1 (0.54) CYP11B1CYP11B2CXCR1CXCR2HTT
SCHEMBL17079612 0.79 MEN1 (0.67) CYP11B1CYP11B2HTTMEN1KMT2A
SCHEMBL17796962 0.77 PTGDR2 (0.49) CXCR1CXCR2HTTMEN1KMT2A
SCHEMBL29450620 0.75 HTT (0.59) HTTMETKDRMEN1KMT2A
SCHEMBL30420875 0.75 CXCR2 (0.50) CXCR1CXCR2HTTMEN1KMT2A
SCHEMBL10665495 0.74 RAB9A (0.79) HTTMEN1KMT2AMAPTLMNA
SCHEMBL10552692 0.74 KDM4E (0.62) CYP11B1CYP11B2KDRMEN1KMT2A
SCHEMBL8946928 0.73 TAAR1 (0.60) HTTMAPTGSK3AGSK3BTSHR
SCHEMBL6165775 0.72 MAPT (0.68) CXCR1CXCR2HTTKDRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US claimed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP claimed
US-5547966-A Aryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-20 US disclosed
EP-0656350-A1 Biaryl urea and related compounds BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-07 EP disclosed