SCHEMBL8970804

SCHEMBL8970804

CCOC(OCC)P(=O)(OCC)C(CC)CC#N

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.33
TSHR P16473 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9140413 0.81 ACHE (0.34) ACHETSHRL3MBTL1MEN1CYP1A2
SCHEMBL7710940 0.77 ACHE (0.38) ACHETSHRL3MBTL1
SCHEMBL8971318 0.75 MEN1 (0.45) TSHRL3MBTL1MEN1CYP1A2KMT2A
SCHEMBL9142655 0.70 NPC1 (0.37) L3MBTL1MEN1KMT2A
SCHEMBL22034591 0.69 TSHR (0.36) TSHRL3MBTL1MEN1CYP1A2KMT2A
SCHEMBL3842819 0.66 ACHE (0.35) ACHETSHRL3MBTL1MEN1CYP1A2
SCHEMBL271779 0.65 THRB (0.38) TSHR
SCHEMBL10343591 0.64 MEN1 (0.38) ACHETSHRL3MBTL1MEN1CYP1A2
SCHEMBL7715865 0.63 ACHE (0.39) ACHETSHRL3MBTL1
Butane SCHEMBL7710937 0.63 FDPS (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5567840-A AS 4-AMINOBUTYRIC ACID AGONIST; MUSCLE RELAXANTS CIBA-GEIGY CORPORATION (US) 1996-10-22 US disclosed
US-5461040-A Therapy of spinal spacticity, multiple sclerosis, cerebral palsy, trigeminus neuralgia, drug withdrawal, pain CIBA-GEIGY CORPORATION (US) 1995-10-24 US disclosed
EP-0399949-B1 Substituted aminoalkylphosphinic acids CIBA GEIGY AG (CH) 1995-04-12 EP disclosed
US-5281747-A Pharmaceuticals CIBA-GEIGY CORPORATION (US) 1994-01-25 US disclosed
EP-0399949-A1 Substituted aminoalkylphosphinic acids CIBA-GEIGY AG (CH) 1990-11-28 EP disclosed