SCHEMBL8971090

SCHEMBL8971090

O=C1C2CCCCC2C(=O)N1C(CCc1ccccc1)C1CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
SLC6A4 P31645 3/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A3 Q01959 2/20 0.39
ALPL P05186 1/20 0.39
GBA1 P04062 1/20 0.37
ACE P12821 6/20 0.36
GABRA1 P14867 3/20 0.36
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
POLB P06746 1/20 0.36
CASR P41180 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9427633 0.89 ALDH1A1 (0.45) ALDH1A1SLC6A4SLC6A2SLC6A3ALPL
SCHEMBL8971016 0.82 TDP1 (0.41) ALDH1A1SLC6A4SLC6A2SLC6A3GBA1
SCHEMBL9428075 0.75 ALDH1A1 (0.41) ALDH1A1SLC6A4SLC6A2SLC6A3ALPL
SCHEMBL493666 0.72 MC4R (0.48) SLC6A4SLC6A2SLC6A3GBA1KMT2A
SCHEMBL8969997 0.69 GBA1 (0.47) SLC6A4SLC6A2SLC6A3GBA1
SCHEMBL7875085 0.69 GBA1 (0.47) SLC6A4SLC6A2SLC6A3GBA1KMT2A
SCHEMBL9978780 0.69 GBA1 (0.47) SLC6A4SLC6A2SLC6A3GBA1
SCHEMBL9428081 0.69 ACHE (0.45) ALDH1A1ACE
SCHEMBL27536629 0.69 CPN1 (0.53) SLC6A4SLC6A2SLC6A3GBA1L3MBTL1
SCHEMBL1101922 0.68 ALDH1A1 (0.70) ALDH1A1KMT2AL3MBTL1CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5480892-A SIGMA RECEPTOR ANTAGONISTS; TREATMENT OF PHYSIOLOGICAL OR DRUG INDUCED PSYCHOSIS AND DYSKINESIA THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-02 US disclosed
US-5356906-A (N-phthalimidoalkyl) piperidines useful as treatments for psychosis THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-10-18 US disclosed
WO-1993022310-A1 (N-PHTHALIMIDOALKYL)PIPERIDINES FOR THE TREATMENT OF PSYCHOSES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-11-11 WO disclosed
WO-1991006297-A1 (N-PHTHALIMIDOALKYL) PIPERIDINES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-05-16 WO disclosed