SCHEMBL8971859

SCHEMBL8971859

Fc1ccc(-c2ccc(C3OCCO3)cc2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.48
CYP11B1 P15538 4/20 0.48
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CCNB2 O95067 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
GSK3B P49841 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
KDM1A O60341 2/20 0.39
CYP17A1 P05093 2/20 0.39
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867644 0.84 MEN1 (0.43) CYP11B2CYP11B1MEN1KMT2ACCNB2
SCHEMBL19509080 0.84 CYP11B1 (0.43) CYP11B2CYP11B1MEN1KMT2ACCNB2
SCHEMBL8972574 0.79 CYP11B2 (0.36) CYP11B2CYP11B1KDM1ACYP17A1RAB9A
SCHEMBL8972569 0.79 CYP11B2 (0.36) CYP11B2CYP11B1KDM1ACYP17A1RAB9A
SCHEMBL19850827 0.79 CYP11B1 (0.47) CYP11B2CYP11B1MEN1KMT2ACCNB2
SCHEMBL19824546 0.77 CYP11B1 (0.43) CYP11B2CYP11B1MEN1KMT2ACYP3A4
SCHEMBL20310639 0.77 CYP11B1 (0.43) CYP11B2CYP11B1MEN1KMT2ACYP3A4
SCHEMBL8972512 0.77 CYP11B2 (0.33) CYP11B2CYP11B1MEN1KMT2AKDM1A
SCHEMBL9312426 0.77 CYP11B2 (0.33) CYP11B2CYP11B1MEN1KMT2AKDM1A
SCHEMBL8972505 0.77 CYP11B2 (0.33) CYP11B2CYP11B1MEN1KMT2AKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433836-B1 Halophenyl substituted dioxanes HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5322638-A Halophenyl substituted dioxanes HOFFMANN-LA ROCHE INC. (US) 1994-06-21 US disclosed
EP-0433836-A2 Halophenyl substituted dioxanes F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed