SCHEMBL8972978

SCHEMBL8972978

COC=C(C(=O)O)c1cccc2ccc(C#CC(O)c3ccccc3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 1/20 0.43
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP2D6 P10635 1/20 0.37
MTNR1A P48039 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
AKR1C3 P42330 1/20 0.32
IKBKE Q14164 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
MTNR1B P49286 1/20 0.31
KMT2A Q03164 1/20 0.31
TACR3 P29371 1/20 0.31
AKR1B1 P15121 1/20 0.31
CACNA2D1 P54289 1/20 0.31
CACNB2 Q08289 1/20 0.31
CACNA1C Q13936 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8972398 0.87 AKR1C2 (0.43) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8972907 0.85 AKR1C2 (0.48) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8961310 0.82 AKR1C2 (0.43) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8973400 0.82 AKR1C2 (0.45) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8972368 0.80 AKR1C2 (0.43) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8626809 0.79 AKR1C2 (0.44) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL4159791 0.79 AKR1C2 (0.44) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8972774 0.79 AKR1C2 (0.42) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8972920 0.79 AKR1C2 (0.43) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL8972800 0.78 AKR1C2 (0.42) AKR1C2CYP3A4CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0566455-B1 Derivatives of 7-ethynyle alpha-(methoxymethylene)1-naphthalenacetic acid, their process of preparation and their use as pesticides ROUSSEL UCLAF (FR) 1996-03-06 EP disclosed
US-5451696-A Parasiticide intermediate ROUSSEL-UCLAF (FR) 1995-09-19 US disclosed
US-5380883-A Insecticide, nematocide, miticide ROUSSEL-UCLAF (FR) 1995-01-10 US disclosed
EP-0566455-A1 Derivatives of 7-ethynyle alpha-(methoxymethylene)1-naphthalenacetic acid, their process of preparation and their use as pesticides ROUSSEL UCLAF (FR) 1993-10-20 EP disclosed