SCHEMBL8973202

SCHEMBL8973202

CCC(C)OC(=O)c1ccc(Cl)cn1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.50
GABRG2 P18507 3/20 0.50
GABRB3 P28472 3/20 0.50
GABRA5 P31644 3/20 0.50
GABRA3 P34903 3/20 0.50
GABRA2 P47869 3/20 0.50
GABRA6 Q16445 1/20 0.50
MAOB P27338 1/20 0.43
TRPA1 O75762 1/20 0.43
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9092992 0.83 GABRA1 (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL4985552 0.78 TRPA1 (0.41) MAOBTRPA1MAPK1L3MBTL1MAPT
SCHEMBL2414269 0.78 CYP1A2 (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31235495 0.78 CYP1A2 (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9155382 0.77 MAPK1 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
Methane SCHEMBL27317936 0.76 CYP1A2 (0.50) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL25612575 0.76 USP2 (0.58) L3MBTL1MAPTTSHR
SCHEMBL12780420 0.75 MAOB (0.51) MAOBTRPA1MAPK1L3MBTL1MAPT
SCHEMBL769167 0.75 MAPK1 (0.65) MAOBTRPA1MAPK1L3MBTL1
SCHEMBL31368564 0.75 MAPK1 (0.65) MAOBTRPA1MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534635-A Process for preparing pyridine-2-carboxamides HOFFMANN-LA ROCHE INC. (US) 1996-07-09 US disclosed
US-5380861-A Process for preparing pyridine 2-carboxamides HOFFMANN-LA ROCHE INC. (US) 1995-01-10 US disclosed