SCHEMBL8973698

SCHEMBL8973698

O=C(O)CN1CCCN(CC(=O)O)CCN(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CCCN(CC(=O)O)CC1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP2 O75604 5/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
TACR1 P25103 4/20 0.51
CYP3A4 P08684 6/20 0.50
CYP2D6 P10635 5/20 0.50
TSHR P16473 4/20 0.50
CASP1 P29466 1/20 0.49
CASP5 P51878 1/20 0.49
HPGD P15428 1/20 0.48
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 2/20 0.48
GAA P10253 1/20 0.48
HIF1A Q16665 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TP53 P04637 1/20 0.46
ACHE P22303 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974312 1.00 USP2 (0.52) USP2CYP1A2CYP2C19TACR1CYP3A4
SCHEMBL8973991 0.96 USP2 (0.56) USP2CYP1A2CYP2C19TACR1CYP3A4
SCHEMBL8973966 0.95 USP2 (0.48) USP2CYP1A2CYP2C19TACR1CYP3A4
SCHEMBL9409753 0.87 TACR1 (0.45) USP2CYP1A2CYP2C19TACR1CYP3A4
SCHEMBL8974017 0.86 ALDH1A1 (0.60) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL8973914 0.86 TACR1 (0.49) TACR1CYP3A4CYP2D6TSHR
SCHEMBL8973982 0.84 HIF1A (0.50) USP2TACR1CYP3A4ALDH1A1KDM4E
SCHEMBL8973968 0.83 USP2 (0.47) USP2CYP1A2TACR1CYP3A4CYP2D6
SCHEMBL6028265 0.81 ALDH1A1 (0.67) USP2CYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL2930604 0.81 USP2 (0.59) USP2CYP1A2CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536491-A 19 F poly aza macrocyclic MRI contrast medium TERUMO KABUSHIKI KAISHA (JP) 1996-07-16 US disclosed
EP-0628316-A1 19F-MRI contrast medium, having a macrocyclic complexant moiety TERUMO KABUSHIKI KAISHA (JP) 1994-12-14 EP disclosed