SCHEMBL9409753

SCHEMBL9409753

NC(=O)C(O)CO.NC(=O)C(O)CO.NC(=O)C(O)CO.O=C(O)CN1CCCN(CC(=O)O)CCN(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)CCCN(CC(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.45
USP2 O75604 6/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 5/20 0.41
TSHR P16473 4/20 0.41
CYP2D6 P10635 4/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CASP1 P29466 1/20 0.40
CASP5 P51878 1/20 0.40
HPGD P15428 1/20 0.39
CYP2C9 P11712 1/20 0.39
HIF1A Q16665 1/20 0.39
MGLL Q99685 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973698 0.87 USP2 (0.52) TACR1USP2CYP1A2CYP2C19CYP3A4
SCHEMBL8974312 0.87 USP2 (0.52) TACR1USP2CYP1A2CYP2C19CYP3A4
SCHEMBL8973991 0.83 USP2 (0.56) TACR1USP2CYP1A2CYP2C19CYP3A4
SCHEMBL8973966 0.83 USP2 (0.48) TACR1USP2CYP1A2CYP2C19CYP3A4
SCHEMBL9409749 0.76 FPR2 (0.50) TACR1USP2CYP1A2CYP2C19CYP3A4
SCHEMBL8974017 0.75 ALDH1A1 (0.60) USP2CYP1A2CYP2C19CYP3A4TSHR
SCHEMBL8973914 0.75 TACR1 (0.49) TACR1CYP3A4TSHRCYP2D6
SCHEMBL8973982 0.73 HIF1A (0.50) TACR1USP2CYP3A4ALDH1A1HIF1A
SCHEMBL8973968 0.72 USP2 (0.47) TACR1USP2CYP1A2CYP3A4TSHR
SCHEMBL6028265 0.71 ALDH1A1 (0.67) USP2CYP1A2CYP2C19CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628316-A1 19F-MRI contrast medium, having a macrocyclic complexant moiety TERUMO KABUSHIKI KAISHA (JP) 1994-12-14 EP disclosed