SCHEMBL8973802

SCHEMBL8973802

CCc1ccc2cccc(OCOC)c2c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
CYP2A6 P11509 1/20 0.44
HTR1B P28222 10/20 0.38
HTR1D P28221 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
SLC6A4 P31645 1/20 0.36
HRH1 P35367 1/20 0.36
TSHR P16473 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25629899 0.83 CYP1A2 (0.50) CYP1A2CYP2A6ALDH1A1MAPT
SCHEMBL18053268 0.81 CYP2A6 (0.50) CYP1A2CYP2A6HTR1BHTR1DALDH1A1
SCHEMBL7129651 0.81 HTR1B (0.40) HTR1BHTR1DMAPTSLC6A4HRH1
SCHEMBL27489770 0.79 HTR2A (0.49) CYP1A2CYP2A6
SCHEMBL8974397 0.78 HTR1B (0.56) CYP1A2HTR1BHTR1DALDH1A1SLC6A4
SCHEMBL29937036 0.78 HTR1B (0.56) CYP1A2HTR1BHTR1DALDH1A1SLC6A4
SCHEMBL8399146 0.74 AKT1 (0.47) CYP1A2CYP2A6ALDH1A1GAAMAPT
SCHEMBL15345486 0.73 HTR1B (0.44) CYP2A6HTR1BALDH1A1GAAMAPT
SCHEMBL1050592 0.73 KDM1A (0.44) HTR1BHTR1DSLC6A4HRH1
SCHEMBL1051243 0.73 KDM1A (0.44) HTR1BHTR1DALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527948-A SUBSTITUTED NAPHTHYL-ALKENOIC ACIDS FOR TREATING AUTOIMMUNE DISORDERS EISAI CORP. LTD. (JP) 1996-06-18 US disclosed
CN-1027064-C Naphthalene derivatives EISAI CO LTD (JP) 1994-12-21 CN disclosed
US-5298649-A Antiinflammatory agents, rheumatic agents and treatment of autoimmune diseases EISAI CO., LTD. (JP) 1994-03-29 US disclosed
EP-0376288-B1 Naphthalene derivative EISAI CO LTD (JP) 1994-03-09 EP disclosed
US-5134111-A Inhibitors of interleukin-1 as antiinflammatory agents EISAI CO., LTD. (JP) 1992-07-28 US disclosed
CN-1043696-A NAPHTHALENE DERIVATIVES EISAI CO LTD (JP) 1990-07-11 CN disclosed
EP-0376288-A1 Naphthalene derivative Eisai Co., Ltd. (JP) 1990-07-04 EP disclosed