SCHEMBL8974107

SCHEMBL8974107

NS(=O)(=O)c1ccc(C2=CCC=C2c2cccnc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.69
CA9 Q16790 9/20 0.69
CA12 O43570 6/20 0.69
CA1 P00915 5/20 0.69
CA4 P22748 1/20 0.49
CA7 P43166 1/20 0.49
DYRK1A Q13627 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
KMT2A Q03164 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
PTGS2 P35354 5/20 0.45
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974347 0.85 PTGS2 (0.62) CA2CA9CA12CA1PTGS2
SCHEMBL8974581 0.83 CA2 (0.57) CA2CA9CA12CA1KMT2A
SCHEMBL8974782 0.82 CA2 (0.68) CA2CA9CA12CA1CA4
SCHEMBL9117865 0.80 CA2 (0.61) CA2CA9CA12CA1CA4
SCHEMBL9130312 0.79 CA9 (0.46) CA2CA9CA12CA1PTGS2
SCHEMBL9114935 0.77 PTGS2 (0.44) CA2CA9CA12CA1CA4
SCHEMBL8658259 0.77 CA2 (0.69) CA2CA9CA12CA1CA4
SCHEMBL8973868 0.76 CA2 (0.48) CA2CA9CA12CA1CA4
SCHEMBL8974243 0.76 CA2 (0.71) CA2CA9CA12CA1CA4
SCHEMBL8974195 0.75 CA9 (0.53) CA2CA9CA12CA1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed