SCHEMBL8974133

SCHEMBL8974133

NS(=O)(=O)c1ccc(C2=CC(CF)(CF)C=C2c2ccc(C(F)(F)F)nc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.43
KCNH2 Q12809 3/20 0.43
MAP4K4 O95819 1/20 0.43
PIK3CA P42336 1/20 0.43
MINK1 Q8N4C8 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
PTGS2 P35354 8/20 0.41
PTGS1 P23219 7/20 0.41
DRD1 P21728 1/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA1 P00915 1/20 0.39
CA4 P22748 1/20 0.39
CA5A P35218 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
PDPK1 O15530 3/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974140 0.89 KCNH2 (0.44) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8974214 0.89 KCNH2 (0.44) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8974342 0.87 KCNH2 (0.54) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974492 0.86 PTGS2 (0.43) PTGS2PTGS1DRD1CA2CA9
SCHEMBL8974393 0.85 KIF11 (0.46) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8973824 0.84 PTGS2 (0.46) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8974138 0.84 KIF11 (0.45) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8973766 0.84 KIF11 (0.64) KIF11PTGS2PTGS1CA2CA9
SCHEMBL9115734 0.83 PTGS2 (0.47) KIF11KCNH2MAP4K4PIK3CAMINK1
SCHEMBL8974199 0.82 KIF11 (0.48) KIF11PTGS2PTGS1DRD1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed