SCHEMBL8974140

SCHEMBL8974140

CCC1(CC)C=C(c2ccc(S(N)(=O)=O)cc2)C(c2ccc(C(F)(F)F)nc2)=C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.44
MAP4K4 O95819 1/20 0.44
PIK3CA P42336 1/20 0.44
MINK1 Q8N4C8 1/20 0.44
PI4KB Q9UBF8 1/20 0.44
PTGS2 P35354 10/20 0.43
PTGS1 P23219 9/20 0.43
KIF11 P52732 1/20 0.42
PDPK1 O15530 5/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 2/20 0.38
CA5A P35218 2/20 0.38
CA9 Q16790 2/20 0.38
CA5B Q9Y2D0 2/20 0.38
PTGES O14684 1/20 0.38
HDAC3 O15379 1/20 0.38
CA12 O43570 1/20 0.38
PDE5A O76074 1/20 0.38
ABCB11 O95342 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974133 0.89 KIF11 (0.43) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974482 0.89 KCNH2 (0.54) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974214 0.88 KCNH2 (0.44) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974376 0.86 PTGS2 (0.45) PTGS2PTGS1CA1CA2CA4
SCHEMBL8973824 0.86 PTGS2 (0.46) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974424 0.84 KIF11 (0.62) PTGS2PTGS1KIF11PDPK1CA1
SCHEMBL8974393 0.84 KIF11 (0.46) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974138 0.83 KIF11 (0.45) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL9118758 0.82 KIF11 (0.47) PTGS2PTGS1KIF11PDPK1CA1
SCHEMBL9115734 0.82 PTGS2 (0.47) KCNH2MAP4K4PIK3CAMINK1PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed