SCHEMBL8974147

SCHEMBL8974147

CC1C=C(c2ccc(S(N)(=O)=O)cc2)C(c2ccc(F)cn2)=C1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.45
CA2 P00918 6/20 0.43
CA1 P00915 4/20 0.43
CA9 Q16790 3/20 0.43
CA5A P35218 3/20 0.43
CA5B Q9Y2D0 3/20 0.43
CA4 P22748 2/20 0.43
PTGS1 P23219 5/20 0.43
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974356 0.92 CA2 (0.43) PTGS2CA2CA1CA9CA5A
SCHEMBL8974495 0.88 CA2 (0.44) PTGS2CA2CA1CA9CA5A
SCHEMBL8974225 0.88 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL8974159 0.86 PTGS2 (0.43) PTGS2CA2CA1CA9CA5A
SCHEMBL8974762 0.86 CA2 (0.42) PTGS2CA2CA1CA9CA5A
SCHEMBL8974183 0.85 CA2 (0.41) PTGS2CA2CA1CA9CA5A
SCHEMBL8974373 0.85 PTGS2 (0.57) PTGS2CA2CA1CA9CA4
SCHEMBL8974071 0.84 CA2 (0.41) PTGS2CA2CA1CA9CA5A
SCHEMBL8974301 0.84 PTGS2 (0.43) PTGS2CA2CA1CA9CA5A
SCHEMBL8974487 0.84 KIF11 (0.50) PTGS2CA2CA1CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed