SCHEMBL8974228

SCHEMBL8974228

NS(=O)(=O)c1ccc(C2=CC(CF)C=C2c2ccc(C(F)(F)F)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.48
PTGS2 P35354 8/20 0.41
PTGS1 P23219 3/20 0.41
CYP2C9 P11712 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
PDPK1 O15530 1/20 0.38
CHRNA7 P36544 2/20 0.37
KDM1A O60341 1/20 0.37
MAOB P27338 1/20 0.37
GCK P35557 1/20 0.36
GCKR Q14397 1/20 0.36
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
MAPT P10636 1/20 0.36
CA4 P22748 2/20 0.36
CA7 P43166 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974181 0.93 KIF11 (0.48) KIF11PTGS2PTGS1CYP2C9PDPK1
SCHEMBL8974259 0.90 KIF11 (0.47) KIF11PTGS2PTGS1CYP2C9KDM4E
SCHEMBL8974933 0.90 KIF11 (0.47) KIF11PTGS2PTGS1CYP2C9KDM4E
SCHEMBL8973758 0.89 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL8974121 0.87 KIF11 (0.51) KIF11PTGS2PTGS1CYP2C9KDM4E
SCHEMBL8974748 0.87 CA2 (0.41) PTGS2PTGS1MAOBCA12CA1
SCHEMBL8974079 0.87 KIF11 (0.64) KIF11PTGS2PTGS1CYP2C9PDPK1
SCHEMBL8974632 0.86 KIF11 (0.50) KIF11PTGS2PTGS1CYP2C9KDM4E
SCHEMBL8973900 0.86 KIF11 (0.50) KIF11PTGS2PTGS1CYP2C9KDM4E
SCHEMBL8974330 0.84 PTGS2 (0.45) KIF11PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed