SCHEMBL8974240

SCHEMBL8974240

NS(=O)(=O)c1ccc(C2=CC(CO)(CO)C=C2c2ccc(Cl)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.59
PTGS1 P23219 4/20 0.59
CA1 P00915 6/20 0.55
CA2 P00918 6/20 0.55
CA9 Q16790 6/20 0.55
CA12 O43570 5/20 0.55
CA4 P22748 2/20 0.55
CA3 P07451 1/20 0.55
CA6 P23280 1/20 0.55
CA5A P35218 1/20 0.55
CA7 P43166 1/20 0.55
CA13 Q8N1Q1 1/20 0.55
CA14 Q9ULX7 1/20 0.55
CA5B Q9Y2D0 1/20 0.55
IKBKB O14920 2/20 0.48
CHUK O15111 2/20 0.48
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
CHRNA7 P36544 1/20 0.47
MEN1 O00255 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973810 0.85 PTGS2 (0.55) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974391 0.85 PTGS2 (0.59) PTGS2PTGS1MAOB
SCHEMBL8973851 0.85 PTGS2 (0.59) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974954 0.85 PTGS2 (0.55) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974325 0.84 CA2 (0.50) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973750 0.81 KIF11 (0.62) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974261 0.80 CA2 (0.60) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974824 0.80 CA2 (0.60) PTGS2PTGS1CA1CA2CA9
SCHEMBL8973866 0.78 PTGS2 (0.48) PTGS2PTGS1CA1CA2CA9
SCHEMBL8974214 0.77 KCNH2 (0.44) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed