SCHEMBL8974245

SCHEMBL8974245

CCC1C=C(c2ccc(F)cc2)C(c2ccc(S(N)(=O)=O)cc2)=C1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.51
PTGS1 P23219 11/20 0.51
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
SOS1 Q07889 1/20 0.46
CHRNA7 P36544 3/20 0.44
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
CA12 O43570 2/20 0.44
CA1 P00915 2/20 0.43
CA7 P43166 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974749 0.86 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8974838 0.86 PTGS2 (0.53) PTGS2PTGS1MAOAMAOBSOS1
SCHEMBL8974405 0.86 CA1 (0.41) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974159 0.86 PTGS2 (0.43) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8973747 0.85 PTGS2 (0.55) PTGS2PTGS1MAOAMAOBSOS1
SCHEMBL8974445 0.84 KIF11 (0.62) PTGS2PTGS1CHRNA7CA2CA9
SCHEMBL8973845 0.84 PTGS2 (0.42) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974373 0.83 PTGS2 (0.57) PTGS2PTGS1MAOAMAOBSOS1
SCHEMBL8974276 0.81 CA1 (0.39) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974080 0.81 PTGS2 (0.57) PTGS2PTGS1MAOAMAOBSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed