SCHEMBL8974445

SCHEMBL8974445

CCC1C=C(c2ccc(C(F)(F)F)cc2)C(c2ccc(S(N)(=O)=O)cc2)=C1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.62
PTGS2 P35354 7/20 0.52
PTGS1 P23219 3/20 0.52
CA12 O43570 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 2/20 0.46
CA1 P00915 2/20 0.46
MAPT P10636 1/20 0.46
CHRNA7 P36544 1/20 0.45
CYP2C9 P11712 1/20 0.44
PDPK1 O15530 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.40
CA7 P43166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974079 0.87 KIF11 (0.64) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974074 0.87 PTGS2 (0.54) KIF11PTGS2
SCHEMBL8974206 0.87 KIF11 (0.47) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974933 0.87 KIF11 (0.47) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974579 0.86 KIF11 (0.62) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974108 0.84 KCNH2 (0.44) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8973917 0.84 KIF11 (0.68) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974245 0.84 PTGS2 (0.51) PTGS2PTGS1CA12CA2CA9
SCHEMBL8974637 0.82 KIF11 (0.70) KIF11PTGS2PTGS1CA12CA2
SCHEMBL8974163 0.82 KIF11 (0.40) KIF11PTGS2PTGS1CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed