SCHEMBL8974266

SCHEMBL8974266

CSc1ccc(C2=CCC=C2c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.62
PTGS1 P23219 4/20 0.46
AKR1C3 P42330 1/20 0.43
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974635 0.85 CA2 (0.47) PTGS2PTGS1TSHR
SCHEMBL2991047 0.82 PTGS2 (0.67) PTGS2PTGS1AKR1C3TSHR
SCHEMBL8974890 0.81 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8974499 0.81 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8974446 0.81 PTGS2 (0.47) PTGS2PTGS1AKR1C3
SCHEMBL9118551 0.80 PTGS2 (0.68) PTGS2PTGS1AKR1C3TSHR
SCHEMBL8974296 0.79 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL8974060 0.79 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8974192 0.79 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL8974390 0.78 PTGS2 (0.47) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed