SCHEMBL8974192

SCHEMBL8974192

CS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(I)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.44
PTGS1 P23219 8/20 0.44
ABCB11 O95342 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MT-CO2 P00403 1/20 0.40
HTR1A P08908 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
MC4R P32245 1/20 0.40
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974499 0.84 PTGS2 (0.61) PTGS2PTGS1ABCB11ALDH1A1MT-CO2
SCHEMBL8974890 0.84 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8974446 0.84 PTGS2 (0.47) PTGS2PTGS1ENPP2
SCHEMBL8974060 0.82 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL8974296 0.82 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL8973815 0.82 CA2 (0.52) PTGS2PTGS1
SCHEMBL8974453 0.81 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL8974390 0.81 PTGS2 (0.47) PTGS2PTGS1ALDH1A1
SCHEMBL514275 0.80 ENPP2 (0.56) PTGS2ENPP2
SCHEMBL8974141 0.79 PTGS2 (0.62) PTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed